Salicylate-urea-based soluble epoxide hydrolase inhibitors with high metabolic and chemical stabilities.
نویسندگان
چکیده
We investigated N-adamantyl-N'-phenyl urea derivatives as simple sEH inhibitors. Salicylate ester derivatives have high inhibitory activities against human sEH, while the free benzoic acids are less active. The methyl salicylate derivative is a potent sEH inhibitor, which also has high metabolic and chemical stabilities; suggesting that such inhibitors are potential lead molecule for bioactive compounds acting in vivo.
منابع مشابه
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Inhibitors of soluble epoxide hydrolase (sEH) represent one of the novel pharmaceutical approaches for treating hypertension, vascular inflammation, pain and other cardiovascular related diseases. Most of the potent sEH inhibitors reported in literature often suffer from poor solubility and bioavailability. Toward improving pharmacokinetic profile beside favorable potency, two series of 4-benza...
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ورودعنوان ژورنال:
- Bioorganic & medicinal chemistry letters
دوره 19 6 شماره
صفحات -
تاریخ انتشار 2009